Tedalinab

Catalog No.: A14189

CB2 receptor agonist

Tedalinab

Tedalinab Chemical Structure

CAS NO. 916591-01-0

Tedalinab (GRC-10693) is a drug developed for the treatment of osteoarthritis and neuropathic pain, which acts as a potent and selective cannabinoid CB2 receptor agonist. It has a very high selectivity of 4700x for CB2 over the related CB1 receptor, has good oral bioavailability and has shown promising safety results and effective analgesic and antiinflammatory actions in early clinical trials.

Availability: In stock

Package Price Qty
5 mg
$220.00
10 mg
$500.00
25 mg
$900.00
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Biological Activity

Tedalinab (GRC-10693) is a drug developed for the treatment of osteoarthritis and neuropathic pain, which acts as a potent and selective cannabinoid CB2 receptor agonist. It has a very high selectivity of 4700x for CB2 over the related CB1 receptor, has good oral bioavailability and has shown promising safety results and effective analgesic and antiinflammatory actions in early clinical trials.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.95 mL 144.76 mL 289.52 mL
0.5 mM 5.79 mL 28.95 mL 57.9 mL
1 mM 2.9 mL 14.48 mL 28.95 mL
5 mM 0.58 mL 2.9 mL 5.79 mL

*The above data is based on the productmolecular weight 345.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14189
Actions Agonist
CAS No. 916591-01-0
Formula C19H21F2N3O
M. Wt 345.4
Solubility DMSO
Purity >98%
Synonyms GRC-10693
SMILES CC(C)(C)NC(=O)C1=NN(C2=C1[[email protected]]3CC[[email protected]@H]2C3)C4=C(C=C(C=C4)F)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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