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Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM.
Targets
| Dipeptidyl peptidase-4 | DPP-9 | DPP-8 | FAP | |
| 1.75 nM | 150 nM | 189 nM | >10 μM |
| In vitro | DMSO | 85 mg/mL (135.16 mM) | |
| Water | 85 mg/mL (135.16 mM) | ||
| Ethanol | 14 mg/mL | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 7.95 mL | 39.75 mL | 79.51 mL |
| 0.5 mM | 1.59 mL | 7.95 mL | 15.9 mL |
| 1 mM | 0.8 mL | 3.98 mL | 7.95 mL |
| 5 mM | 0.16 mL | 0.8 mL | 1.59 mL |
*The above data is based on the productmolecular weight 1257.72. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A15258 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 906093-29-6 |
| Formula | C44H65Br5N12O2S2 |
| M. Wt | 1257.72 |
| Purity | >98% |
| SMILES | CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.Br.Br.Br.Br.Br |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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