Teneligliptin hydrobromide

Catalog No.: A15258

DPP-4 inhibitor

Teneligliptin hydrobromide

Teneligliptin hydrobromide Chemical Structure

CAS NO. 906093-29-6

Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM.

Availability: In stock

Package Price Qty
100 mg
$240.00
200 mg
$440.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM.
Targets
Dipeptidyl peptidase-4 DPP-9 DPP-8 FAP
1.75 nM150 nM189 nM>10 μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 7.95 mL 39.75 mL 79.51 mL
0.5 mM 1.59 mL 7.95 mL 15.9 mL
1 mM 0.8 mL 3.98 mL 7.95 mL
5 mM 0.16 mL 0.8 mL 1.59 mL

*The above data is based on the productmolecular weight 1257.72. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15258
Actions Inhibitor
M. Wt 1257.72
Formula C44H65Br5N12O2S2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 906093-29-6
Synonyms N/A
SMILES CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.Br.Br.Br.Br.Br

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