TM38837 is a selective inverse agonist targeting cannabinoid receptor 1 (CB1), exhibiting an IC50 of 24 nM. With a significantly higher selectivity for CB1 over cannabinoid receptor 2 (CB2) (IC50: 4500 nM), TM38837 demonstrates potential in modulating metabolic processes. Its biological activity includes reducing body weight and improving plasma inflammatory markers and glucose homeostasis, making it a valuable tool for research on metabolic disorders and obesity.
TM38837 is a selective inverse agonist targeting cannabinoid receptor 1 (CB1), exhibiting an IC50 of 24 nM. With a significantly higher selectivity for CB1 over cannabinoid receptor 2 (CB2) (IC50: 4500 nM), TM38837 demonstrates potential in modulating metabolic processes. Its biological activity includes reducing body weight and improving plasma inflammatory markers and glucose homeostasis, making it a valuable tool for research on metabolic disorders and obesity.
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