Tolvaptan

Catalog No.: A11594

vasopressin receptor 2 antagonist

Tolvaptan Chemical Structure

CAS NO. 150683-30-0

Tolvaptan is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28μM.

Availability: In stock

Package Price Qty
5 mg
$70.00
10 mg
$120.00
25 mg
$240.00
50 mg
$380.00
10mM * 1mL in DMSO
$120.00

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Biological Activity

Tolvaptan is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28μM.
Targets
vasopressin receptor 2 vasopressin receptor 1a
3 nM580 nM
In vitro DMSO 90 mg/mL (200.47 mM)
Water <1 mg/mL (<1 mM)
Ethanol 6 mg/mL (13.36 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.27 mL 111.37 mL 222.75 mL
0.5 mM 4.45 mL 22.27 mL 44.55 mL
1 mM 2.23 mL 11.14 mL 22.27 mL
5 mM 0.45 mL 2.23 mL 4.45 mL

*The above data is based on the productmolecular weight 448.94. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11594
Actions Antagonist
M. Wt 448.94
Formula C26H25ClN2O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 150683-30-0
SMILES CC1=CC=CC=C1C(=O)NC2=CC(=C(C=C2)C(=O)N3CCCC(C4=C3C=CC(=C4)Cl)O)C

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