TX1-85-1

Catalog No.: A16361

Her3 (ErbB3) ligand

TX1-85-1

TX1-85-1 Chemical Structure

CAS NO. 1603845-32-4

TX1-85-1 is ErbB3 inhibitor. TX2-121-1 may exert Her3-dependent pharmacology through an allosteric mechanismthereby disrupting interactions between Her3 and other proteins such as Her3 or cMet consistent with results presented here and distinct from conventional kinase inhibitors, which block catalytic function.

Availability: In stock

Package Price Qty
5 mg
$160.00
10 mg
$300.00
50 mg
$900.00
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Biological Activity

TX1-85-1 is ErbB3 inhibitor. TX2-121-1 may exert Her3-dependent pharmacology through an allosteric mechanismthereby disrupting interactions between Her3 and other proteins such as Her3 or cMet consistent with results presented here and distinct from conventional kinase inhibitors, which block catalytic function.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.22 mL 86.1 mL 172.21 mL
0.5 mM 3.44 mL 17.22 mL 34.44 mL
1 mM 1.72 mL 8.61 mL 17.22 mL
5 mM 0.34 mL 1.72 mL 3.44 mL

*The above data is based on the productmolecular weight 580.69. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16361
Actions Inhibitor
CAS No. 1603845-32-4
Formula C32H36N8O3
M. Wt 580.69
Solubility DMSO
Purity >98%
Synonyms TX1 85-1, TX185-1, TX1851, TX 1851, TX-1851
SMILES C=CC(NC1=CC(C2=NN(C3CCC(N4CCN(C(C)=O)CC4)CC3)C5=NC=NC(N)=C52)=CC=C1OC6=CC=CC=C6)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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