Vortioxetine (Lu AA21004) hydrobromide

Catalog No.: A12602

5-HT Receptor modulator

Vortioxetine (Lu AA21004) hydrobromide

Vortioxetine (Lu AA21004) hydrobromide Chemical Structure

CAS NO. 960203-27-4

Lu-AA21004 is an oral multimodal serotonergic agent, inhibits 5-HT(1A), 5-HT(1B), 5-HT(3A), 5-HT(7) and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.

Availability: In stock

Package Price Qty
5 mg
$70.00
10 mg
$110.00
25 mg
$280.00
50 mg
$150.00
10mM * 1mL in DMSO
$77.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Lu-AA21004 is an oral multimodal serotonergic agent, inhibits 5-HT(1A), 5-HT(1B), 5-HT(3A), 5-HT(7) and SERT with IC50 of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively.
Targets
SERT 5-HT3A 5-HT1A 5-HT7 5-HT1B
1.6 nM(Ki)3.7 nM(Ki)15 nM(Ki)19 nM(Ki)33 nM(Ki)
In vitro (25°C) DMSO 76 mg/mL (200.33 mM)
Water <1 mg/mL (<1 mM)
Ethanol 17 mg/mL (44.81 mM)
In vivo 15% Captisol, pH 9 10 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.36 mL 131.8 mL 263.6 mL
0.5 mM 5.27 mL 26.36 mL 52.72 mL
1 mM 2.64 mL 13.18 mL 26.36 mL
5 mM 0.53 mL 2.64 mL 5.27 mL

*The above data is based on the productmolecular weight 379.36. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12602
Actions Modulator
M. Wt 379.36
Formula C18H22N2S.HBr
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 960203-27-4
Synonyms Lu AA21004, LuAA21004, Lu-AA21004
SMILES CC1=CC(=C(C=C1)SC2=CC=CC=C2N3CCNCC3)C.Br

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