WDR5-0103

Catalog No.: A15928

WDR5 antagonist

WDR5-0103

WDR5-0103 Chemical Structure

CAS NO. 890190-22-4

WDR5-0103 is a small molecule that binds a peptide-binding pocket on WDR5 (Kd = 450 nM), inhibiting the catalytic activity of the MLL core complex in vitro (IC50 = 39 M).

Availability: In stock

Package Price Qty
10 mg

Regular Price: $90.00

Special Price $72.00

25 mg

Regular Price: $200.00

Special Price $160.00

50 mg

Regular Price: $350.00

Special Price $280.00

Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

WDR5-0103 is a small molecule that binds a peptide-binding pocket on WDR5 (Kd = 450 nM), inhibiting the catalytic activity of the MLL core complex in vitro (IC50 = 39 M).
In vitro DMSO 68 mg/mL (177.34 mM)
Water Insoluble
Ethanol 18 mg/mL (46.94 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.08 mL 130.4 mL 260.79 mL
0.5 mM 5.22 mL 26.08 mL 52.16 mL
1 mM 2.61 mL 13.04 mL 26.08 mL
5 mM 0.52 mL 2.61 mL 5.22 mL

*The above data is based on the productmolecular weight 383.45. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15928
Actions Antagonist
CAS No. 890190-22-4
Formula C21H25N3O4
M. Wt 383.45
Purity >98%
Synonyms WDR 5-0103, WDR-5-0103
SMILES O=C(OC)C1=CC(NC(C2=CC=CC(OC)=C2)=O)=C(N3CCN(C)CC3)C=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy WDR5-0103 | WDR5-0103 Supplier | purchase | cost | manufacturer | order | distributor | buy 890190-22-4| 890190-22-4 Supplier | purchase 890190-22-4 | 890190-22-4 cost | 890190-22-4 manufacturer | order 890190-22-4 | 890190-22-4 distributor
Rewards