WDR5-0103

Catalog No.: A15928

WDR5 antagonist

WDR5-0103 Chemical Structure

CAS NO. 890190-22-4

WDR5-0103 is a small molecule that binds a peptide-binding pocket on WDR5 (Kd = 450 nM), inhibiting the catalytic activity of the MLL core complex in vitro (IC50 = 39 M).

Availability: In stock

Package Price Qty
10 mg
$90.00
25 mg
$200.00
50 mg
$350.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

WDR5-0103 is a small molecule that binds a peptide-binding pocket on WDR5 (Kd = 450 nM), inhibiting the catalytic activity of the MLL core complex in vitro (IC50 = 39 M).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.08 mL 130.4 mL 260.79 mL
0.5 mM 5.22 mL 26.08 mL 52.16 mL
1 mM 2.61 mL 13.04 mL 26.08 mL
5 mM 0.52 mL 2.61 mL 5.22 mL

*The above data is based on the productmolecular weight 383.45. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15928
Actions Antagonist
M. Wt 383.45
Formula C21H25N3O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 890190-22-4
Synonyms WDR 5-0103, WDR-5-0103
SMILES O=C(OC)C1=CC(NC(C2=CC=CC(OC)=C2)=O)=C(N3CCN(C)CC3)C=C1

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