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YM-1758735

Catalog No.: A85026
Androgen Receptor Antagonist
YM-1758735 is an orally active androgen receptor (AR) antagonist that exhibits an IC50 of 0.2 μM. This compound effectively inhibits AR-mediated transcriptional activation, making it a valuable tool for studying androgen signaling pathways. YM-1758735 is particularly relevant for research focused on prostate cancer and other androgen-related disorders.
YM-1758735 262294-30-4 Androgen Receptor Antagonist
Grouped product items
Size Price Stock Qty
25mg
$1,275.00
In stock
50mg
$1,625.00
In stock
100mg
$2,000.00
In stock
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Free Delivery on orders over $500
Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionYM-1758735 is an orally active androgen receptor (AR) antagonist that exhibits an IC50 of 0.2 μM. This compound effectively inhibits AR-mediated transcriptional activation, making it a valuable tool for studying androgen signaling pathways. YM-1758735 is particularly relevant for research focused on prostate cancer and other androgen-related disorders.
Product Information
Catalog NumA85026
FormulaC21H19F5N4O
Molecular Weight438.40
CAS Number262294-30-4
SMILESC[C@@H]1N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C[C@@H](C)N(C(NC3=C(F)C=C(F)C=C3)=O)C1
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Endocrinology-Hormones > Androgen Receptors