Ziritaxestat
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | Ziritaxestat (GLPG1690) is a first-in-class autotaxin (ATX) inhibitor, with an IC50 of 131 nM and Ki of 15 nM. | ||
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Targets |
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Catalog Num | A19312 |
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Formula | C30H33FN8O2S |
Molecular Weight | 588.7 |
CAS Number | 1628260-79-6 |
SMILES | N#CC1=C(C2=CC=C(F)C=C2)N=C(N(C3=C(CC)N=C4C(C)=CC(N5CCN(CC(N6CC(O)C6)=O)CC5)=CN43)C)S1 |
Synonyms | GLPG1690, GLPG-1690, GLPG 1690 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 87 mg/mL (147.78 mM) | |
Water | Insoluble | ||
Ethanol | 3 mg/mL (5.09 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 16.99 mL | 84.93 mL | 169.87 mL |
0.5 mM | 3.4 mL | 16.99 mL | 33.97 mL |
1 mM | 1.7 mL | 8.49 mL | 16.99 mL |
5 mM | 0.34 mL | 1.7 mL | 3.4 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2