1-Azakenpaullone

Catalog No.: A14303

GSK-3β inhibitor

1-Azakenpaullone Chemical Structure

CAS NO. 676596-65-9

1-Azakenpaullone is a potent and selective GSK-3β inhibitor with IC50 of 18 nM, >100-fold selectivity over CDK1/cyclin B and CDK5/p25.

Availability: In stock

Package Price Qty
2 mg
$120.00
5 mg
$237.00
10 mg
$360.00
10mM * 1mL in DMSO
$256.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

1-Azakenpaullone is a potent and selective GSK-3β inhibitor with IC50 of 18 nM, >100-fold selectivity over CDK1/cyclin B and CDK5/p25.
Targets
GSK-3α GSK-3β
In vitro DMSO 66 mg/mL (201.12 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.47 mL 152.36 mL 304.73 mL
0.5 mM 6.09 mL 30.47 mL 60.95 mL
1 mM 3.05 mL 15.24 mL 30.47 mL
5 mM 0.61 mL 3.05 mL 6.09 mL

*The above data is based on the productmolecular weight 328.16. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14303
Actions Inhibitor
M. Wt 328.16
Formula C15H10BrN3O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 676596-65-9
Synonyms N/A
SMILES C1C2=C(C3=C(C=CC=N3)NC1=O)NC4=C2C=C(C=C4)Br

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