1-Azakenpaullone

Catalog No.: A14303

GSK-3β inhibitor

1-Azakenpaullone

1-Azakenpaullone Chemical Structure

CAS NO. 676596-65-9

1-Azakenpaullone is a potent and selective GSK-3β inhibitor with IC50 of 18 nM, >100-fold selectivity over CDK1/cyclin B and CDK5/p25.

Availability: In stock

Package Price Qty
2 mg

Regular Price: $120.00

Special Price $96.00

5 mg

Regular Price: $237.00

Special Price $189.60

10 mg

Regular Price: $360.00

Special Price $288.00

10mM * 1mL in DMSO

Regular Price: $256.00

Special Price $204.80

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Biological Activity

1-Azakenpaullone is a potent and selective GSK-3β inhibitor with IC50 of 18 nM, >100-fold selectivity over CDK1/cyclin B and CDK5/p25.
Targets
GSK-3α GSK-3β
In vitro DMSO 58 mg/mL (176.74 mM)
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.47 mL 152.36 mL 304.73 mL
0.5 mM 6.09 mL 30.47 mL 60.95 mL
1 mM 3.05 mL 15.24 mL 30.47 mL
5 mM 0.61 mL 3.05 mL 6.09 mL

*The above data is based on the productmolecular weight 328.16. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14303
Actions Inhibitor
CAS No. 676596-65-9
Formula C15H10BrN3O
M. Wt 328.16
Purity >98%
SMILES C1C2=C(C3=C(C=CC=N3)NC1=O)NC4=C2C=C(C=C4)Br
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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