3BrB-PP1

Catalog No.: A55209
ATP Analog
3BrB-PP1 is an ATP-competitive analog designed to selectively inhibit protein kinases with mutations in the ATP-binding pocket, particularly targeting the Thr97 mutation within Sty1. This compound offers a unique tool for investigating the effects of ATP-binding site alterations on kinase activity. Its specificity makes it valuable for studying mutant forms of kinases in various biological contexts and cancer research.
Grouped product items
Size Price Stock Qty
5mg
$345.00
In stock
10mg
$530.00
In stock
25mg
$1,060.00
In stock
50mg
$1,550.00
In stock
100mg
$2,240.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

Loading distributor info...

Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
Description3BrB-PP1 is an ATP-competitive analog designed to selectively inhibit protein kinases with mutations in the ATP-binding pocket, particularly targeting the Thr97 mutation within Sty1. This compound offers a unique tool for investigating the effects of ATP-binding site alterations on kinase activity. Its specificity makes it valuable for studying mutant forms of kinases in various biological contexts and cancer research.
Product Information
Catalog NumA55209
FormulaC16H18BrN5
Molecular Weight360.25
CAS Number956025-99-3
SMILESNC1=C2C(N(C(C)(C)C)N=C2CC3=CC=CC(Br)=C3)=NC=N1
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2