5-HT6 Inverse Agonist 1 is a selective antagonist of the 5-HT6 receptor, exhibiting a Ki of 23 nM and a Kb of 6.62 nM. This compound effectively inhibits the 5-HT6R-mediated signaling pathways, including Cdk5 and mTOR. Additionally, 5-HT6 Inverse Agonist 1 has demonstrated efficacy in reducing tactile hypersensitivity in a rat model of spinal nerve ligation, making it a valuable tool for research into pain management and neurobiology.
5-HT6 Inverse Agonist 1 is a selective antagonist of the 5-HT6 receptor, exhibiting a Ki of 23 nM and a Kb of 6.62 nM. This compound effectively inhibits the 5-HT6R-mediated signaling pathways, including Cdk5 and mTOR. Additionally, 5-HT6 Inverse Agonist 1 has demonstrated efficacy in reducing tactile hypersensitivity in a rat model of spinal nerve ligation, making it a valuable tool for research into pain management and neurobiology.
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