A-1165442

Catalog No.: A21516

TRPV1 antagonist

A-1165442

A-1165442 Chemical Structure

CAS NO. 1221443-94-2

A-1165442 is a potent, competitive and orally available TRPV1 antagonist with an IC50 of 9 nM for human TRPV1.

Availability: In stock

Package Price Qty
1 mg
$162.00
5 mg
$486.00
10 mg
$828.00
50 mg
$2,484.00
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Biological Activity

A-1165442 is a potent, competitive and orally available TRPV1 antagonist with an IC50 of 9 nM for human TRPV1.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.16 mL 115.78 mL 231.56 mL
0.5 mM 4.63 mL 23.16 mL 46.31 mL
1 mM 2.32 mL 11.58 mL 23.16 mL
5 mM 0.46 mL 2.32 mL 4.63 mL

*The above data is based on the productmolecular weight 431.86. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21516
Actions Antagonist
CAS No. 1221443-94-2
Formula C22H20ClF2N3O2
M. Wt 431.86
Purity >98%
Synonyms A1165442, A 1165442
SMILES O=C(NC1=CC=CC2=C1C=C(C)N=C2)N[[email protected]]3C4=CC=C(Cl)C=C4OC(CF)(CF)C3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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