A-438079 HCl

Catalog No.: A12597

P2X7 receptor antagonist

A-438079 HCl

A-438079 HCl Chemical Structure

CAS NO. 899507-36-9

A-438079 HCl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line). Devoid of activity at other P2 receptors (IC50 >> 10 uM).

Availability: In stock

Package Price Qty
5 mg
$85.00
10 mg
$130.00
50 mg
$380.00
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Biological Activity

A-438079 HCl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line). Devoid of activity at other P2 receptors (IC50 >> 10 uM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.19 mL 145.94 mL 291.88 mL
0.5 mM 5.84 mL 29.19 mL 58.38 mL
1 mM 2.92 mL 14.59 mL 29.19 mL
5 mM 0.58 mL 2.92 mL 5.84 mL

*The above data is based on the productmolecular weight 342.608. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12597
Actions Antagonist
CAS No. 899507-36-9
Formula C13H10Cl3N5
M. Wt 342.608
Purity >98%
Synonyms A-438079 , A 438079, A438079, A-438079 HCl
SMILES ClC1=CC=CC(C2=NN=NN2CC3=CN=CC=C3)=C1Cl.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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