A 438079 hydrochloride

Catalog No.: A14983

P2X7 receptor antagonist

A 438079 hydrochloride

A 438079 hydrochloride Chemical Structure

CAS NO. 899431-18-6

A 438079 Hcl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line).

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10 mg
$95.00
25 mg
$215.00
50 mg
$395.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Zhihua Yi, .et al. Andrographolide Inhibits Mechanical and Thermal Hyperalgesia in a Rat Model of HIV-Induced Neuropathic Pain, Front Pharmacol, 2018, 9: 593 PMID: 29950989

Biological Activity

A 438079 Hcl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line).
Targets
P2X7 receptor
6.9(pIC50)
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.19 mL 145.94 mL 291.88 mL
0.5 mM 5.84 mL 29.19 mL 58.38 mL
1 mM 2.92 mL 14.59 mL 29.19 mL
5 mM 0.58 mL 2.92 mL 5.84 mL

*The above data is based on the productmolecular weight 342.61. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14983
Actions Antagonist
M. Wt 342.61
Formula C13H10Cl3N5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 899431-18-6
SMILES C1=CC(=C(C(=C1)Cl)Cl)C2=NN=NN2CC3=CN=CC=C3.Cl

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