Acetyl-Calpastatin (184-210) (human)

Catalog No.: A15290

Selective calpain inhibitor

Acetyl-Calpastatin (184-210) (human) Chemical Structure

CAS NO. 123714-50-1

Acetyl-Calpastatin (184-210) (human), selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 uM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.

Availability: In stock

Package Price Qty
1 mg
$235.00
5 mg
$635.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Acetyl-Calpastatin (184-210) (human), selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 uM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 3.15 mL 15.73 mL 31.47 mL
0.5 mM 0.63 mL 3.15 mL 6.29 mL
1 mM 0.31 mL 1.57 mL 3.15 mL
5 mM 0.06 mL 0.31 mL 0.63 mL

*The above data is based on the productmolecular weight 3177.65. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15290
Actions Inhibitor
M. Wt 3177.65
Formula C142H230N36O44S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 123714-50-1
Synonyms N/A
SMILES CC[[email protected]](C)[[email protected]](NC(=O)[[email protected]](CC1=CC=C(O)C=C1)NC(=O)[[email protected]@H](NC(=O)[[email protected]](CO)NC(=O)[[email protected]](CO)NC(=O)[[email protected]](CCSC)NC(=O)[[email protected]@H]1CCCN1C(=O)[[email protected]](CC(O)=O)NC(C)=O)[[email protected]@H](C)O)C(=O)N[[email protected]@H](CCC(O)=O)C(=O)N[[email protected]@H](CCC(O)=O)C(=O)N[[email protected]@H](CC(C)C)C(=O)NCC(=O)N[[email protected]@H](CCCCN)C(=O)N[[email protected]@H](CCCNC(N)=N)C(=O)N[[email protected]@H](CCC(O)=O)C(=O)N[[email protected]@H](C(C)C)C(=O)N[[email protected]@H]([[email protected]@H](C)O)C(=O)N[[email protected]@H]([[email protected]@H](C)CC)C(=O)N1CCC[[email protected]]1C(=O)N1CCC[[email protected]]1C(=O)N[[email protected]@H](CCCCN)C(=O)N[[email protected]@H](CC1=CC=C(O)C=C1)C(=O)N[[email protected]@H](CCCNC(N)=N)C(=O)N[[email protected]@H](CCC(O)=O)C(=O)N[[email protected]@H](CC(C)C)C(=O)N[[email protected]@H](CC(C)C)C(=O)N[[email protected]@H](C)C(N)=O

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