AM095 free base

Catalog No.: A14180

LPA1 Receptor antagonist

AM095 free base

AM095 free base Chemical Structure

CAS NO. 1228690-36-5

AM095 is a novel, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 0.73 and 0.98 μM for mouse or recombinant human LPA1, respectively

Availability: Out of stock

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5 mg
$100.00
10 mg
$140.00
25 mg
$270.00
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Biological Activity

AM095 is a novel, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 0.73 and 0.98 μM for mouse or recombinant human LPA1, respectively
In vitro DMSO 84 mg/mL (184.01 mM)
Water Insoluble
Ethanol 3 mg/mL (6.57 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.91 mL 109.53 mL 219.06 mL
0.5 mM 4.38 mL 21.91 mL 43.81 mL
1 mM 2.19 mL 10.95 mL 21.91 mL
5 mM 0.44 mL 2.19 mL 4.38 mL

*The above data is based on the productmolecular weight 456.49. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14180
Actions Antagonist
CAS No. 1228690-36-5
Formula C27H24N2O5
M. Wt 456.49
Solubility DMSO
Purity >98%
Synonyms AM 095,AM-095
SMILES CC1=NOC(=C1NC(=O)O[[email protected]](C)C2=CC=CC=C2)C3=CC=C(C=C3)C4=CC=C(C=C4)CC(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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