LPA Receptor

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  1. LPA Receptor Antagonist

    Ki16425 is a LPA receptor antagonist with selectivity for LPA1 and LPA3 and exhibits Ki values of 0.34, 6.5, and 0.93 μM for the human LPA1, LPA2, and LPA3 receptors, respectively.
  2. LPA Receptor antagonist

    Ki16198 is a potent LPA receptor antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively.
  3. lysophaphatidic acid 1 (LPA1/Edg-2) receptor inhibitor

    SAR-100842 is a lysophaphatidic acid 1 (LPA1/Edg-2) receptor inhibitor.
  4. LPA1 receptor antagonist

    AM095 is a potent LPA1 receptor antagonist because it inhibited GTP??S binding to Chinese hamster ovary (CHO) cell membranes overexpressing recombinant human or mouse LPA1 with IC50 values of 0.98 and 0.73 μM, respectively, and exhibited no LPA1 agonism.
  5. LPA1 receptor antagonist

    AM966 is a high affinity, selective, oral antagonist of LPA1 receptor (lysophosphatidic acid receptor) with an IC50 value of 17 nM.
  6. LPA1 Receptor antagonist

    AM095 is a novel, potent and orally bioavailable antagonist of lysophosphatidic acid type 1 receptor (LPA1) with IC50 values of 0.73 and 0.98 μM for mouse or recombinant human LPA1, respectively
  7. LPA2 agonist

    GRI 977143, selective lysophosphatidic acid 2 (LPA2) receptor non-lipid agonist (EC50 = 3.3 uM).
  8. LPA1 antagonist

    ONO-7300243 is a novel, potent lysophosphatidic acid receptor 1 (LPA1) antagonist with IC50 of 0.16 μM.
  9. LPA2 agonist

    Radioprotectin-1 is a potent and specific nonlipid agonist of lysophosphatidic acid receptor 2 (LPA2), with an EC50 value of 25 nM for murine LPA2 subtype.
  10. LPA5 antagonist

    AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia.
  11. LPA1 receptor antagonist

    ASP6432 is a potent and selective Type 1 Lysophosphatidic Acid (LPA1) receptor antagonist.
  12. LPA1 antagonist

    BMS-986020 is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist.
  13. LPA1 antagonist

    LPA1 antagonist 1 is a highly selective Lysophosphatidic Acid receptor-1 (LPA1) antagonist with an IC50 of 25 nM.
  14. LPA2 antagonist

    LPA2 antagonist 1 is a LPA2 antagonist with an IC50 of 17 nM.
  15. LPA1 antagonist

    BMS-986020 sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist.

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