AM211

Catalog No.: A21612

PGD2) receptor type 2 (DP2) antagonist

AM211

AM211 Chemical Structure

CAS NO. 1175526-27-8

AM211 is a potent, selective and orally bioavailable prostaglandin D2 (PGD2) receptor type 2 (DP2) antagonist, with IC50s of 4.9 nM, 7.8 nM, 4.9 nM, 10.4 nM for human, mouse, guinea pig, and rat DP2, respectively.

Availability: In stock

Package Price Qty
5 mg
$81.00
10 mg
$140.00
50 mg
$414.00
100 mg
$828.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

AM211 is a potent, selective and orally bioavailable prostaglandin D2 (PGD2) receptor type 2 (DP2) antagonist, with IC50s of 4.9 nM, 7.8 nM, 4.9 nM, 10.4 nM for human, mouse, guinea pig, and rat DP2, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.98 mL 99.9 mL 199.8 mL
0.5 mM 4 mL 19.98 mL 39.96 mL
1 mM 2 mL 9.99 mL 19.98 mL
5 mM 0.4 mL 2 mL 4 mL

*The above data is based on the productmolecular weight 500.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21612
Actions Antagonist
CAS No. 1175526-27-8
Formula C27H27F3N2O4
M. Wt 500.51
Solubility DMSO
Purity >98%
Synonyms AM211 free acid, AM 211, AM-211
SMILES O=C(O)CC1=CC(C2=CC=C(C(F)(F)F)C=C2CN(CC)C(NCC3=CC=CC=C3)=O)=C(OC)C=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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