AS2717638

Catalog No.: A18630

LPA5 antagonist

AS2717638

AS2717638 Chemical Structure

CAS NO. 2148339-28-8

AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia.

Availability: In stock

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5 mg
$420.00
10 mg
$700.00
50 mg
$2,100.00
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Biological Activity

AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.35 mL 111.74 mL 223.47 mL
0.5 mM 4.47 mL 22.35 mL 44.69 mL
1 mM 2.23 mL 11.17 mL 22.35 mL
5 mM 0.45 mL 2.23 mL 4.47 mL

*The above data is based on the productmolecular weight 447.48. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18630
Actions Antagonist
M. Wt 447.48
Formula C25H25N3O5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2148339-28-8
Synonyms AS 2717638, AS-2717638
SMILES O=C1N(C2=NOC3=C2C=C(C)C=C3)C=C(C(N4CCCCC4)=O)C5=C1C=C(OC)C(OC)=C5

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