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BIM-23027

Catalog No.: A60143
sst2 Receptor Agonist
BIM-23027 is a selective agonist of the sst2 receptor, exhibiting an EC50 of 0.32 nM. This compound mimics the action of somatostatin (SRIF), a cyclic tetradecapeptide, and plays a critical role in stimulating dopamine release through a Glu-dependent mechanism. BIM-23027 is suitable for research applications focusing on neuroendocrine regulation and receptor pharmacology.
BIM-23027 78981-49-4 sst2 Receptor Agonist
Grouped product items
Size Price Stock Qty
1mg
$40.00
In stock
5mg
$100.00
In stock
10mg
$170.00
In stock
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Free Delivery on orders over $500
Research use only. We do not sell to patients.
Data Sheet SDS

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionBIM-23027 is a selective agonist of the sst2 receptor, exhibiting an EC50 of 0.32 nM. This compound mimics the action of somatostatin (SRIF), a cyclic tetradecapeptide, and plays a critical role in stimulating dopamine release through a Glu-dependent mechanism. BIM-23027 is suitable for research applications focusing on neuroendocrine regulation and receptor pharmacology.
Product Information
Catalog NumA60143
FormulaC43H54N8O7
Molecular Weight794.94
CAS Number78981-49-4
Sequence shorteningCyclo[{(NMe)Ala}-FWKTF]
SMILESC(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@H](C)N(C)C(=O)[C@H](CC5=CC=CC=C5)NC(=O)[C@]([C@@H](C)O)(NC(=O)[C@H](CCCCN)NC3=O)[H]
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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GPCR/G Protein > Somatostatin Receptors