Somatostatin Receptors

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  1. somatostatin receptor antagonist

    Octreotide is a peptide agonist for sst2, sst3 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: 290 - 1140 (sst1), 0.4 - 2.1 (sst2), 4.4 - 34.5 (sst3), > 1000 (sst4), and 5.6 - 32 (sst5).
  2. Somatostatin is an endogenous peptide noted to inhibit the release of growth hormone, insulin and glucagon.
  3. somatostatin receptor 2 antagonist

    CYN-154806 is a potent selective somatostatin receptor 2 (sst2) antagonist.
  4. Somatostatin receptors agonist

    Pasireotide(SOM 230) is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively).
  5. SSTR5 antagonist

    SSTR5 Antagonist 1 (compound 10) is a highly potent, oral active and selective somatostatin (receptor) subtype 5 (SSTR5) antagonist and has potential to treat type 2 diabetes mellitus (T2DM).
  6. somatostatin receptor 2 antagonist

    DOTA-JR11 is a somatostatin receptor 2 ??SSTR2??antagonist. DOTA-JR11 can be labeled by 68Ga, used for paired imaging in neuroendocrine tumors (NETs) research.

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