BNS808 is a selective antagonist of the cannabinoid-1 receptor (CB1R), demonstrating an IC50 value of 0.8 nM while exhibiting notable selectivity for the CB2 receptor and limited central nervous system penetration. This compound is primarily utilized in research focused on obesity and its related metabolic disorders, including metabolic dysfunction-associated steatotic liver disease (MASLD). BNS808's reduced availability for CNS entry enhances its safety profile and minimizes the potential for drug-drug interactions due to high plasma protein binding.
BNS808 is a selective antagonist of the cannabinoid-1 receptor (CB1R), demonstrating an IC50 value of 0.8 nM while exhibiting notable selectivity for the CB2 receptor and limited central nervous system penetration. This compound is primarily utilized in research focused on obesity and its related metabolic disorders, including metabolic dysfunction-associated steatotic liver disease (MASLD). BNS808's reduced availability for CNS entry enhances its safety profile and minimizes the potential for drug-drug interactions due to high plasma protein binding.
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