Cariprazine-d8 is a deuterated form of Cariprazine, a novel antipsychotic agent primarily targeting dopamine D3 and D2 receptors with high affinities of Ki = 0.085 nM and Ki = 0.49 nM, respectively. It also shows moderate affinity for the serotonin receptor 5-HT1A (Ki = 2.6 nM). This stable isotope-labeled compound enables enhanced pharmacokinetic studies and metabolic profiling in research applications, contributing valuable insights into therapeutic mechanisms and drug interactions.
Cariprazine-d8 is a deuterated form of Cariprazine, a novel antipsychotic agent primarily targeting dopamine D3 and D2 receptors with high affinities of Ki = 0.085 nM and Ki = 0.49 nM, respectively. It also shows moderate affinity for the serotonin receptor 5-HT1A (Ki = 2.6 nM). This stable isotope-labeled compound enables enhanced pharmacokinetic studies and metabolic profiling in research applications, contributing valuable insights into therapeutic mechanisms and drug interactions.
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