CCG215022

Catalog No.: A16189

GRK2/5 inhibitor

CCG215022 Chemical Structure

CAS NO. 1813527-81-9

CCG215022 is a potent GRK2 and GRK5 inhibitor. CCG215022 exhibited nanomolar IC50 values against both GRK2 and GRK5 and good selectivity against other closely related kinases such as GRK1 and PKA.

Availability: In stock

Package Price Qty
1 mg
$120.00
5 mg
$320.00
10 mg
$480.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CCG215022 is a potent GRK2 and GRK5 inhibitor. CCG215022 exhibited nanomolar IC50 values against both GRK2 and GRK5 and good selectivity against other closely related kinases such as GRK1 and PKA.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.02 mL 100.1 mL 200.2 mL
0.5 mM 4 mL 20.02 mL 40.04 mL
1 mM 2 mL 10.01 mL 20.02 mL
5 mM 0.4 mL 2 mL 4 mL

*The above data is based on the productmolecular weight 499.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16189
Actions Inhibitor
M. Wt 499.51
Formula C26H22FN7O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1813527-81-9
Synonyms CCG 215022, CCG-215022
SMILES O=C(C1=C(F)C=CC(C2C(C(NC3=CC=C(NN=C4)C4=C3)=O)=C(C)NC(N2)=O)=C1)NCC5=NC=CC=C5

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