CCT128930

Catalog No.: A11031

AKT Inhibitor

CCT128930

CCT128930 Chemical Structure

CAS NO. 885499-61-6

CCT128930 is an ATP-competitive AKT inhibitor that is a potent, advanced lead pyrrolopyrimidine compound exhibiting selectivity for AKT over PKA, achieved by targeting a single amino acid difference.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $128.00

Special Price $115.20

25 mg

Regular Price: $256.00

Special Price $230.40

50 mg

Regular Price: $450.00

Special Price $405.00

100 mg

Regular Price: $720.00

Special Price $648.00

10mM * 1mL in DMSO

Regular Price: $103.00

Special Price $92.70

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CCT128930 is an ATP-competitive AKT inhibitor that is a potent, advanced lead pyrrolopyrimidine compound exhibiting selectivity for AKT over PKA, achieved by targeting a single amino acid difference.
Targets
Akt2 (Cell-free assay) p70 S6K (Cell-free assay) PKA (Cell-free assay)
6 nM120 nM168 nM
In vitro (25°C) DMSO 68 mg/mL (198.92 mM)
Water <1 mg/mL (<1 mM)
Ethanol 6 mg/mL (17.55 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 11 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.26 mL 146.28 mL 292.57 mL
0.5 mM 5.85 mL 29.26 mL 58.51 mL
1 mM 2.93 mL 14.63 mL 29.26 mL
5 mM 0.59 mL 2.93 mL 5.85 mL

*The above data is based on the productmolecular weight 341.8 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A11031
Actions Inhibitor
M. Wt 341.8
Formula C18H20ClN5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 885499-61-6
Synonyms CCT-128930
SMILES C1CN(CCC1(CC2=CC=C(C=C2)Cl)N)C3=NC=NC4=C3C=CN4

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
You may also be interested in the following product(s)
Keywords:buy CCT128930 | CCT128930 Supplier | purchase CCT128930 | CCT128930 cost | CCT128930 manufacturer | order CCT128930 | CCT128930 distributor | buy 885499-61-6| 885499-61-6 Supplier | purchase 885499-61-6 | 885499-61-6 cost | 885499-61-6 manufacturer | order 885499-61-6 | 885499-61-6 distributor
Rewards