Total item
Cart Subtotal
$0.00 Biological Activity
CCT137690 is a highly selective inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 15 nM, 25 nM and 19 nM. It has little effect on hERG ion-channel.
Targets
| Aurora A | Aurora C | Aurora B | ||
| 15 nM | 19 nM | 25 nM |
| In vitro (25°C) | DMSO | 4 mg/mL (7.25 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| In vivo | 1% DMSO+30% polyethylene glycol+1% Tween 80 | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 18.13 mL | 90.66 mL | 181.32 mL |
| 0.5 mM | 3.63 mL | 18.13 mL | 36.26 mL |
| 1 mM | 1.81 mL | 9.07 mL | 18.13 mL |
| 5 mM | 0.36 mL | 1.81 mL | 3.63 mL |
*The above data is based on the productmolecular weight 551.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A11081 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1095382-05-0 |
| Formula | C26H31BrN8O |
| M. Wt | 551.5 |
| Purity | >98% |
| Synonyms | CCT-137690 |
| SMILES | CC1=CC(=NO1)CN2CCN(CC2)C3=C4C(=NC=C3Br)N=C(N4)C5=CC=C(C=C5)N6CCN(CC6)C |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy CCT137690 | CCT137690 Supplier | purchase | cost | manufacturer | order | distributor | buy 1095382-05-0| 1095382-05-0 Supplier | purchase 1095382-05-0 | 1095382-05-0 cost | 1095382-05-0 manufacturer | order 1095382-05-0 | 1095382-05-0 distributor
Adooq Quality Guarantee
We promise all products perform as described.