CCT137690

Catalog No.: A11081

Aurora Kinase inhibitor

CCT137690

CCT137690 Chemical Structure

CAS NO. 1095382-05-0

CCT137690 is a highly selective inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 15 nM, 25 nM and 19 nM. It has little effect on hERG ion-channel.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $85.00

Special Price $68.00

10 mg

Regular Price: $110.00

Special Price $88.00

50 mg

Regular Price: $400.00

Special Price $320.00

100 mg

Regular Price: $625.00

Special Price $500.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

CCT137690 is a highly selective inhibitor of Aurora A, Aurora B and Aurora C with IC50 of 15 nM, 25 nM and 19 nM. It has little effect on hERG ion-channel.
Targets
Aurora A Aurora C Aurora B
15 nM19 nM25 nM
In vitro (25°C) DMSO 4 mg/mL (7.25 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.13 mL 90.66 mL 181.32 mL
0.5 mM 3.63 mL 18.13 mL 36.26 mL
1 mM 1.81 mL 9.07 mL 18.13 mL
5 mM 0.36 mL 1.81 mL 3.63 mL

*The above data is based on the productmolecular weight 551.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A11081
Actions Inhibitor
M. Wt 551.5
Formula C26H31BrN8O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1095382-05-0
Synonyms CCT-137690
SMILES CC1=CC(=NO1)CN2CCN(CC2)C3=C4C(=NC=C3Br)N=C(N4)C5=CC=C(C=C5)N6CCN(CC6)C

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