CJ-42794

Catalog No.: A21948

EP4 antagonist

CJ-42794

CJ-42794 Chemical Structure

CAS NO. 847728-01-2

CJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3).

Availability: In stock

Package Price Qty
10 mg
$54.00
25 mg
$108.00
50 mg
$186.00
100 mg
$318.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.16 mL 120.82 mL 241.65 mL
0.5 mM 4.83 mL 24.16 mL 48.33 mL
1 mM 2.42 mL 12.08 mL 24.16 mL
5 mM 0.48 mL 2.42 mL 4.83 mL

*The above data is based on the productmolecular weight 413.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21948
Actions Antagonist
M. Wt 413.83
Formula C22H17ClFNO4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 847728-01-2
Synonyms CJ-042794, CJ042794, CJ 042794; CJ 42794, CJ42794
SMILES ClC1=CC=C(OC2=CC=C(F)C=C2)C(C(N[[email protected]](C3=CC=C(C(O)=O)C=C3)C)=O)=C1

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy CJ-42794 | CJ-42794 Supplier | purchase | cost | manufacturer | order | distributor | buy 847728-01-2| 847728-01-2 Supplier | purchase 847728-01-2 | 847728-01-2 cost | 847728-01-2 manufacturer | order 847728-01-2 | 847728-01-2 distributor
Rewards