CJ-42794

Catalog No.: A21948

EP4 antagonist

CJ-42794

CJ-42794 Chemical Structure

CAS NO. 847728-01-2

CJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3).

Availability: In stock

Package Price Qty
10 mg

Regular Price: $54.00

Special Price $43.20

25 mg

Regular Price: $108.00

Special Price $86.40

50 mg

Regular Price: $186.00

Special Price $148.80

100 mg

Regular Price: $318.00

Special Price $254.40

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Biological Activity

CJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.16 mL 120.82 mL 241.65 mL
0.5 mM 4.83 mL 24.16 mL 48.33 mL
1 mM 2.42 mL 12.08 mL 24.16 mL
5 mM 0.48 mL 2.42 mL 4.83 mL

*The above data is based on the productmolecular weight 413.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21948
Actions Antagonist
CAS No. 847728-01-2
Formula C22H17ClFNO4
M. Wt 413.83
Purity >98%
Synonyms CJ-042794, CJ042794, CJ 042794; CJ 42794, CJ42794
SMILES ClC1=CC=C(OC2=CC=C(F)C=C2)C(C(N[[email protected]](C3=CC=C(C(O)=O)C=C3)C)=O)=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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