CMP8 is a selective ligand for the estrogen receptor, specifically targeting the mutant estrogen receptor ligand binding domain (ERLBD). This compound demonstrates potent biological activity with IC50 values of 29 nM for MGERα, 41 nM for MGRERα, 1100 nM for human ERα, and 2200 nM for human ERβ. CMP8 is valuable for research applications focused on estrogen receptor modulation and its role in cancer biology.
CMP8 is a selective ligand for the estrogen receptor, specifically targeting the mutant estrogen receptor ligand binding domain (ERLBD). This compound demonstrates potent biological activity with IC50 values of 29 nM for MGERα, 41 nM for MGRERα, 1100 nM for human ERα, and 2200 nM for human ERβ. CMP8 is valuable for research applications focused on estrogen receptor modulation and its role in cancer biology.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
