Cyamemazine-d6 is a deuterated derivative of Cyamemazine, a neuroleptic agent characterized by its phenothiazine structure. This compound functions primarily as a potent antagonist of the 5-HT3 (Ki of 12 nM), 5-HT2A (Ki of 1.5 nM), and 5-HT2C (Ki of 75 nM) receptors, exhibiting notable anxiolytic and antipsychotic properties. Cyamemazine-d6 serves as a valuable stable isotope for studies involving pharmacokinetics, trace labeling, and metabolic research in the context of psychiatric disorders.
Cyamemazine-d6 is a deuterated derivative of Cyamemazine, a neuroleptic agent characterized by its phenothiazine structure. This compound functions primarily as a potent antagonist of the 5-HT3 (Ki of 12 nM), 5-HT2A (Ki of 1.5 nM), and 5-HT2C (Ki of 75 nM) receptors, exhibiting notable anxiolytic and antipsychotic properties. Cyamemazine-d6 serves as a valuable stable isotope for studies involving pharmacokinetics, trace labeling, and metabolic research in the context of psychiatric disorders.
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