dBET57

Catalog No.: A19133

BRD4BD1degrader

dBET57

dBET57 Chemical Structure

CAS NO. 1883863-52-2

dBET57 is a potent and selective degrader of BRD4BD1 based on the PROTAC technology.

Availability: In stock

Package Price Qty
5 mg
$120.00
10 mg
$220.00
50 mg
$500.00
100 mg
$800.00
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Biological Activity

dBET57 is a potent and selective degrader of BRD4BD1 based on the PROTAC technology.
In vitro DMSO 89 mg/mL (127.29 mM)
Water Insoluble
Ethanol 11 mg/mL (15.73 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.3 mL 71.51 mL 143.02 mL
0.5 mM 2.86 mL 14.3 mL 28.6 mL
1 mM 1.43 mL 7.15 mL 14.3 mL
5 mM 0.29 mL 1.43 mL 2.86 mL

*The above data is based on the productmolecular weight 699.18. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A19133
Actions Degrader
CAS No. 1883863-52-2
Formula C34H31ClN8O5S
M. Wt 699.18
Solubility DMSO
Purity >98%
Synonyms dBET 57, dBET-57
SMILES O=C(NCCNC1=CC=CC(C(N2C(CC3)C(NC3=O)=O)=O)=C1C2=O)C[[email protected]]4C5=NN=C(C)N5C6=C(C(C)=C(C)S6)C(C7=CC=C(Cl)C=C7)=N4
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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