Deltarasin HCl

Catalog No.: A13722

PDE-KRAS inhibitor

Deltarasin HCl

Deltarasin HCl Chemical Structure

CAS NO. 1440898-61-2

Deltarasin is a novel small molecule inhibiting the KRAS PDEδ interaction and thus impairing oncogenic KRAS signalling.

Availability: In stock

Package Price Qty
5 mg
$150.00
10 mg
$210.00
25 mg
$420.00
10mM * 1mL in DMSO
$195.00
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Biological Activity

Deltarasin is a novel small molecule inhibiting the KRAS PDEδ interaction and thus impairing oncogenic KRAS signalling.
Targets
PDEδ
38 nM(Kd)
In vitro DMSO 89 mg/mL (147.41 mM)
Water Insoluble
Ethanol 89 mg/mL (147.41 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.47 mL 72.33 mL 144.65 mL
0.5 mM 2.89 mL 14.47 mL 28.93 mL
1 mM 1.45 mL 7.23 mL 14.47 mL
5 mM 0.29 mL 1.45 mL 2.89 mL

*The above data is based on the productmolecular weight 691.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13722
Actions Inhibitor
CAS No. 1440898-61-2
Formula C40H37N5O.2.4HCl
M. Wt 691.3
Solubility DMSO
Purity >98%
SMILES C1CNCCC1[[email protected]@H](COC2=CC=C(C=C2)C3=NC4=CC=CC=C4N3CC5=CC=CC=C5)N6C7=CC=CC=C7N=C6C8=CC=CC=C8
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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