Deltarasin HCl

Catalog No.: A13722

PDE-KRAS inhibitor

Deltarasin HCl

Deltarasin HCl Chemical Structure

CAS NO. 1440898-61-2

Deltarasin is a novel small molecule inhibiting the KRAS PDEδ interaction and thus impairing oncogenic KRAS signalling.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $150.00

Special Price $135.00

10 mg

Regular Price: $210.00

Special Price $189.00

25 mg

Regular Price: $420.00

Special Price $378.00

10mM * 1mL in DMSO

Regular Price: $195.00

Special Price $175.50

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Deltarasin is a novel small molecule inhibiting the KRAS PDEδ interaction and thus impairing oncogenic KRAS signalling.
Targets
PDEδ
38 nM(Kd)
In vitro DMSO 100 mg/mL (165.63 mM)
Water <1 mg/mL (<1 mM)
Ethanol 100 mg/mL (165.63 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.47 mL 72.33 mL 144.65 mL
0.5 mM 2.89 mL 14.47 mL 28.93 mL
1 mM 1.45 mL 7.23 mL 14.47 mL
5 mM 0.29 mL 1.45 mL 2.89 mL

*The above data is based on the productmolecular weight 691.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13722
Actions Inhibitor
M. Wt 691.3
Formula C40H37N5O.2.4HCl
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1440898-61-2
Synonyms N/A
SMILES C1CNCCC1[[email protected]@H](COC2=CC=C(C=C2)C3=NC4=CC=CC=C4N3CC5=CC=CC=C5)N6C7=CC=CC=C7N=C6C8=CC=CC=C8

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