Dersimelagon is a selective agonist of the melanocortin 1 receptor (MC1R) with demonstrated efficacy in human (EC50 of 8.16 nM), cynomolgus monkey (3.91 nM), mouse (1.14 nM), and rat (0.251 nM) models. It exhibits strong binding affinity for hMC1R and hMC4R, with Ki values of 2.26 nM and 32.9 nM, respectively. This compound is primarily utilized in research focused on skin pigmentation and the modulation of melanin synthesis.
Dersimelagon is a selective agonist of the melanocortin 1 receptor (MC1R) with demonstrated efficacy in human (EC50 of 8.16 nM), cynomolgus monkey (3.91 nM), mouse (1.14 nM), and rat (0.251 nM) models. It exhibits strong binding affinity for hMC1R and hMC4R, with Ki values of 2.26 nM and 32.9 nM, respectively. This compound is primarily utilized in research focused on skin pigmentation and the modulation of melanin synthesis.
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