Drinabant is a potent antagonist of the CB1 receptor, specifically designed for oral activity. It effectively inhibits agonist-stimulated calcium signaling, demonstrating IC50 values of 25 nM for human CB1 receptors and 10 nM for rat CB1 receptors, while showing no efficacy against human CB2 receptors. This compound is valuable for research applications involving the endocannabinoid system and its role in various physiological processes.
Drinabant is a potent antagonist of the CB1 receptor, specifically designed for oral activity. It effectively inhibits agonist-stimulated calcium signaling, demonstrating IC50 values of 25 nM for human CB1 receptors and 10 nM for rat CB1 receptors, while showing no efficacy against human CB2 receptors. This compound is valuable for research applications involving the endocannabinoid system and its role in various physiological processes.
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