Biological Activity
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 19.96 mL | 99.8 mL | 199.59 mL |
0.5 mM | 3.99 mL | 19.96 mL | 39.92 mL |
1 mM | 2 mL | 9.98 mL | 19.96 mL |
5 mM | 0.4 mL | 2 mL | 3.99 mL |
*The above data is based on the productmolecular weight 501.02. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A21207 |
---|---|
Actions | Antagonist |
CAS No. | 913064-47-8 |
Formula | C29H29ClN4O2 |
M. Wt | 501.02 |
Purity | >98% |
Synonyms | ELN441958, ELN 441958 |
SMILES | ClC1=C2C(CN(C3=CC=CC(C(N4CCC5(CCN(C6=CC=NC=C6)CC5)CC4)=O)=C3)C2=O)=CC=C1 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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