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GPCR/G Protein
Bradykinin Receptor

Bradykinin Receptor

Catalog No.

Product Name

Application

Product Information

Product Citation

A12964

FR167344 free base

nonpeptide bradykinin receptor B2 antagonist

FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist.

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A13839

SSR240612

bradykinin B1 receptor antagonist

SSR240612 is a new antagonist of the bradykinin B1 receptor.

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- Ling Qin, .et al. , Arthritis Res Ther, 2019, 21:12 PMID: 30621761
A18074

Icatibant

Bradykinin B2 receptors antagonist

Icatibant (HOE-140) is a selective and specific antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively.

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A21207

ELN-441958

B1 receptor antagonist

ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.

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A23883

R715

bradykinin B1 receptor antagonist

R715 is a selective bradykinin B1 receptor antagonist. R715 significantly attenuates the hyperalgesic effect developed in Streptozotocin-diabetic mice.

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