Epoxomicin

Catalog No.: A12730

Proteasome inhibitor

Epoxomicin

Epoxomicin Chemical Structure

CAS NO. 134381-21-8

Epoxomicin is a potent anti-tumor agent isolated from Actinomycetes that is used as a selective and irreversible inhibitor of the 20S proteasome.

Availability: In stock

Package Price Qty
2 mg
$120.00
5 mg
$250.00
10 mg
$450.00
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Biological Activity

Epoxomicin is a potent anti-tumor agent isolated from Actinomycetes that is used as a selective and irreversible inhibitor of the 20S proteasome.
Targets
20S proteasome
In vitro DMSO 98 mg/mL (176.66 mM)
Water Insoluble
Ethanol 98 mg/mL (176.66 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.03 mL 90.14 mL 180.28 mL
0.5 mM 3.61 mL 18.03 mL 36.06 mL
1 mM 1.8 mL 9.01 mL 18.03 mL
5 mM 0.36 mL 1.8 mL 3.61 mL

*The above data is based on the productmolecular weight 554.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12730
Actions Inhibitor
CAS No. 134381-21-8
Formula C28H50N4O7
M. Wt 554.7
Solubility DMSO
Purity >98%
Synonyms BU-4061T
SMILES CC[[email protected]](C)[[email protected]@H](NC(=O)[[email protected]]([[email protected]@H](C)CC)N(C)C(=O)C)C(=O)N[[email protected]@H]([[email protected]@H](C)O)C(=O)N[[email protected]](CC(C)C)C(=O)[[email protected]]1(C)OC1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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