ERα degrader-2 is a selective estrogen receptor degrader (SERD) that exhibits potent binding affinity for the estrogen receptor alpha (ERα) with an IC50 of 17.1 nM and demonstrates robust degradation efficacy with an EC50 of 0.3 nM. This compound possesses favorable pharmacokinetic properties, making it a valuable tool for studying HER2-positive breast cancer. ERα degrader-2 is suitable for applications in cancer research, particularly in investigating therapeutic strategies targeting ERα signaling pathways.
ERα degrader-2 is a selective estrogen receptor degrader (SERD) that exhibits potent binding affinity for the estrogen receptor alpha (ERα) with an IC50 of 17.1 nM and demonstrates robust degradation efficacy with an EC50 of 0.3 nM. This compound possesses favorable pharmacokinetic properties, making it a valuable tool for studying HER2-positive breast cancer. ERα degrader-2 is suitable for applications in cancer research, particularly in investigating therapeutic strategies targeting ERα signaling pathways.
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