ERRα antagonist-1 is a selective antagonist of estrogen-related receptor α (ERRα), effectively inhibiting its interaction with coactivators Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, with IC50 values of 170 nM and 180 nM, respectively. This compound is valuable for research applications focused on metabolic regulation and mitochondrial function, providing a tool for exploring ERRα's role in various physiological processes and disease states. ERRα antagonist-1 facilitates investigations into the therapeutic potential of targeting ERRα pathways in metabolic disorders and cancer.
ERRα antagonist-1 is a selective antagonist of estrogen-related receptor α (ERRα), effectively inhibiting its interaction with coactivators Proliferator-activated Receptor γ Coactivator-1α (PGC-1α) and PGC-1β, with IC50 values of 170 nM and 180 nM, respectively. This compound is valuable for research applications focused on metabolic regulation and mitochondrial function, providing a tool for exploring ERRα's role in various physiological processes and disease states. ERRα antagonist-1 facilitates investigations into the therapeutic potential of targeting ERRα pathways in metabolic disorders and cancer.
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