ESI-09

Catalog No.: A14233

EPAC1/EPAC2 inhibitor

ESI-09

ESI-09 Chemical Structure

CAS NO. 263707-16-0

ESI-09 is a specific exchange protein directly activated by cAMP (EPAC) inhibitor with IC50 of 3.2 uM and 1.4 uM for EPAC1 and EPAC2,

Availability: In stock

Package Price Qty
10 mg
$120.00
25 mg
$208.00
50 mg
$400.00
10mM * 1mL in DMSO
$90.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

ESI-09 is a specific exchange protein directly activated by cAMP (EPAC) inhibitor with IC50 of 3.2 uM and 1.4 uM for EPAC1 and EPAC2,
Targets
EPAC2 EPAC1
1.4 μM3.2 μM
In vitro DMSO 66 mg/mL (199.53 mM)
Water <1 mg/mL (<1 mM)
Ethanol 20 mg/mL heating (60.46 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.23 mL 151.16 mL 302.32 mL
0.5 mM 6.05 mL 30.23 mL 60.46 mL
1 mM 3.02 mL 15.12 mL 30.23 mL
5 mM 0.6 mL 3.02 mL 6.05 mL

*The above data is based on the productmolecular weight 330.77. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A14233
Actions Inhibitor
M. Wt 330.77
Formula C16H15ClN4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 263707-16-0
Synonyms 0
SMILES CC(C)(C)C1=CC(=NO1)C(=O)/C(=N/NC2=CC(=CC=C2)Cl)/C#N

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