EZH2-IN-4 is a potent inhibitor of the EZH2 enzyme, exhibiting IC50 values of 0.923 nM for wild type EZH2 and 2.65 nM for mutant EZH2. This compound demonstrates significant anti-cancer activity, making it a valuable tool for research in cancer therapeutics and epigenetic regulation. Its oral bioavailability enhances its potential for in vivo studies targeting EZH2-driven malignancies.
EZH2-IN-4 is a potent inhibitor of the EZH2 enzyme, exhibiting IC50 values of 0.923 nM for wild type EZH2 and 2.65 nM for mutant EZH2. This compound demonstrates significant anti-cancer activity, making it a valuable tool for research in cancer therapeutics and epigenetic regulation. Its oral bioavailability enhances its potential for in vivo studies targeting EZH2-driven malignancies.
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