FR 180204

Catalog No.: A14119

ERK inhibitor

FR 180204

FR 180204 Chemical Structure

CAS NO. 865362-74-9

FR 180204 is a novel and selective inhibitor of extracellular signal-regulated kinase (ERK), which may be a potential new therapy for rheumatoid arthritis.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $120.00

Special Price $108.00

25 mg

Regular Price: $250.00

Special Price $225.00

50 mg

Regular Price: $400.00

Special Price $360.00

10mM * 1mL in DMSO

Regular Price: $95.00

Special Price $85.50

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

FR 180204 is a novel and selective inhibitor of extracellular signal-regulated kinase (ERK), which may be a potential new therapy for rheumatoid arthritis.
Targets
ERK2 ERK1
0.14 μM(Ki)0.31 μM(Ki)
In vitro DMSO 65 mg/mL (198.57 mM)
Water <1 mg/mL (<1 mM)
Ethanol 2 mg/mL heating (6.1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.55 mL 152.75 mL 305.49 mL
0.5 mM 6.11 mL 30.55 mL 61.1 mL
1 mM 3.05 mL 15.27 mL 30.55 mL
5 mM 0.61 mL 3.05 mL 6.11 mL

*The above data is based on the productmolecular weight 327.34. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A14119
Actions Inhibitor
M. Wt 327.34
Formula C18H13N7
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 865362-74-9
Synonyms FR-180204,FR180204
SMILES C1=CC=C(C=C1)C2=NN3C=CC=CC3=C2C4=CC5=C(NN=C5N=N4)N

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy FR 180204 | FR 180204 Supplier | purchase FR 180204 | FR 180204 cost | FR 180204 manufacturer | order FR 180204 | FR 180204 distributor | buy 865362-74-9| 865362-74-9 Supplier | purchase 865362-74-9 | 865362-74-9 cost | 865362-74-9 manufacturer | order 865362-74-9 | 865362-74-9 distributor
Rewards