GGTI298 Trifluoroacetate

Catalog No.: A16560

GGTase I inhibitor

GGTI298 Trifluoroacetate

GGTI298 Trifluoroacetate Chemical Structure

CAS NO. 1217457-86-7

GGTI298 Trifluoroacetate is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor, which can inhibit Rap1A with IC50 of 3 μM; little effect on Ha-Ras with IC50 of >20 μM.

Availability: In stock

Package Price Qty
1 mg
$54.00
5 mg
$162.00
10 mg
$276.00
50 mg
$828.00
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Biological Activity

GGTI298 Trifluoroacetate is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor, which can inhibit Rap1A with IC50 of 3 μM; little effect on Ha-Ras with IC50 of >20 μM.
In vitro DMSO 87 mg/mL (146.54 mM)
Water Insoluble
Ethanol 87 mg/mL (146.54 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.84 mL 84.22 mL 168.45 mL
0.5 mM 3.37 mL 16.84 mL 33.69 mL
1 mM 1.68 mL 8.42 mL 16.84 mL
5 mM 0.34 mL 1.68 mL 3.37 mL

*The above data is based on the productmolecular weight 593.66. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16560
Actions Inhibitor
CAS No. 1217457-86-7
Formula C29H34F3N3O5S
M. Wt 593.66
Solubility DMSO
Purity >98%
Synonyms GGTI 298, GGTI-298
SMILES CC(C)C[[email protected]@H](C(OC)=O)NC(C1=CC=C(NC[[email protected]@H](N)CS)C=C1C2=C3C=CC=CC3=CC=C2)=O.O=C(O)C(F)(F)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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