GGTI298 Trifluoroacetate

Name: GGTI298 Trifluoroacetate
SKU: A16560
Price: 45 USD
Rating: 5 (288 reviews)

Catalog No.: A16560

GGTase I inhibitor

GGTI298 Trifluoroacetate is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor, which can inhibit Rap1A with IC50 of 3 μM; little effect on Ha-Ras with IC50 of >20 μM.

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Grouped product items
Size	Price	Stock
1mg	$45.00	In stock
5mg	$155.00	In stock
10mg	$245.00	In stock
25mg	$485.00	In stock
50mg	$675.00	In stock
*10mM 1mL in DMSO**	$205.00	In stock
Bulk Size	Bulk Discount

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Data Sheet

SDS

Other Forms of GGTI298 Trifluoroacetate

GGTI298

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Biological Activity

Discription	GGTI298 Trifluoroacetate is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor, which can inhibit Rap1A with IC50 of 3 μM; little effect on Ha-Ras with IC50 of >20 μM.

Product Information

Catalog Num	A16560
Formula	C29H34F3N3O5S
Molecular Weight	593.66
CAS Number	1217457-86-7
SMILES	CC(C)C[C@@H](C(OC)=O)NC(C1=CC=C(NC[C@@H](N)CS)C=C1C2=C3C=CC=CC3=CC=C2)=O.O=C(O)C(F)(F)F
Synonyms	GGTI 298, GGTI-298
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro	DMSO	87 mg/mL (146.54 mM)
	Water	Insoluble
	Ethanol	87 mg/mL (146.54 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	16.84 mL	84.22 mL	168.45 mL
0.5 mM	3.37 mL	16.84 mL	33.69 mL
1 mM	1.68 mL	8.42 mL	16.84 mL
5 mM	0.34 mL	1.68 mL	3.37 mL

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