GGTI298 Trifluoroacetate

Catalog No.: A16560

GGTase I inhibitor

GGTI298 Trifluoroacetate

GGTI298 Trifluoroacetate Chemical Structure

CAS NO. 1217457-86-7

GGTI298 Trifluoroacetate is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor, which can inhibit Rap1A with IC50 of 3 μM; little effect on Ha-Ras with IC50 of >20 μM.

Availability: In stock

Package Price Qty
1 mg
$54.00
5 mg
$162.00
10 mg
$276.00
50 mg
$828.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

GGTI298 Trifluoroacetate is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor, which can inhibit Rap1A with IC50 of 3 μM; little effect on Ha-Ras with IC50 of >20 μM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.84 mL 84.22 mL 168.45 mL
0.5 mM 3.37 mL 16.84 mL 33.69 mL
1 mM 1.68 mL 8.42 mL 16.84 mL
5 mM 0.34 mL 1.68 mL 3.37 mL

*The above data is based on the productmolecular weight 593.66. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16560
Actions Inhibitor
M. Wt 593.66
Formula C29H34F3N3O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1217457-86-7
Synonyms GGTI 298, GGTI-298
SMILES CC(C)C[[email protected]@H](C(OC)=O)NC(C1=CC=C(NC[[email protected]@H](N)CS)C=C1C2=C3C=CC=CC3=CC=C2)=O.O=C(O)C(F)(F)F

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy GGTI298 Trifluoroacetate | GGTI298 Trifluoroacetate Supplier | purchase | cost | manufacturer | order | distributor | buy 1217457-86-7| 1217457-86-7 Supplier | purchase 1217457-86-7 | 1217457-86-7 cost | 1217457-86-7 manufacturer | order 1217457-86-7 | 1217457-86-7 distributor
Rewards