GPR81 agonist 2

Catalog No.: A60906
GPR81 Agonist
GPR81 Agonist 2 specifically targets the GPR81 receptor, exhibiting potent agonistic activity with EC50 values of 0.023 µM for human GPR81 and 0.123 µM for human GPR109A. This compound is valuable for research in metabolic regulation, insulin sensitivity, and tumor metabolism. Its ability to selectively activate GPR81 makes it a useful tool for probing signaling pathways related to energy homeostasis and lipid metabolism.
Grouped product items
Size Price Stock Qty
25mg
$2,160.00
In stock
50mg
$2,770.00
In stock
100mg
$3,680.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Nature Volume 622 Issue 7982 (2023)
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Nature volume 574, pages268-272 (2019)
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Biological Activity
DescriptionGPR81 Agonist 2 specifically targets the GPR81 receptor, exhibiting potent agonistic activity with EC50 values of 0.023 µM for human GPR81 and 0.123 µM for human GPR109A. This compound is valuable for research in metabolic regulation, insulin sensitivity, and tumor metabolism. Its ability to selectively activate GPR81 makes it a useful tool for probing signaling pathways related to energy homeostasis and lipid metabolism.
Product Information
Catalog NumA60906
FormulaC26H27ClN6O5S2
Molecular Weight603.11
CAS Number1143024-28-5
SMILESO=C(NC1=NC2=C(S1)C=C(S(=O)(C3CCN(CC3)C)=O)C=C2)NC(C4=C(Cl)C=C(OCC)C(N5N=CC=C5)=C4)=O
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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