GSK1016790A

Catalog No.: A15854

TRPV4 Activator

GSK1016790A

GSK1016790A Chemical Structure

CAS NO. 942206-85-1

GSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells.

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$140.00
25 mg
$280.00
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Biological Activity

GSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells.
Targets
TRPV4
In vitro DMSO 98 mg/mL (149.47 mM)
Water Insoluble
Ethanol 98 mg/mL (149.47 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.25 mL 76.26 mL 152.53 mL
0.5 mM 3.05 mL 15.25 mL 30.51 mL
1 mM 1.53 mL 7.63 mL 15.25 mL
5 mM 0.31 mL 1.53 mL 3.05 mL

*The above data is based on the productmolecular weight 655.61. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15854
Actions Activator
CAS No. 942206-85-1
Formula C28H32Cl2N4O6S2
M. Wt 655.61
Purity >98%
Synonyms GSK101
SMILES CC(C)CC(C(=O)N1CCN(CC1)C(=O)C(CO)NS(=O)(=O)C2=C(C=C(C=C2)Cl)Cl)NC(=O)C3=CC4=CC=CC=C4S3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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