GSK1016790A

Catalog No.: A15854

TRPV4 Activator

GSK1016790A

GSK1016790A Chemical Structure

CAS NO. 942206-85-1

GSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells.

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$140.00
25 mg
$280.00
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Biological Activity

GSK1016790A is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34nM in choroid plexus epithelial cells.
Targets
TRPV4
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.25 mL 76.26 mL 152.53 mL
0.5 mM 3.05 mL 15.25 mL 30.51 mL
1 mM 1.53 mL 7.63 mL 15.25 mL
5 mM 0.31 mL 1.53 mL 3.05 mL

*The above data is based on the productmolecular weight 655.61. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15854
Actions Activator
M. Wt 655.61
Formula C28H32Cl2N4O6S2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 942206-85-1
Synonyms GSK101
SMILES CC(C)CC(C(=O)N1CCN(CC1)C(=O)C(CO)NS(=O)(=O)C2=C(C=C(C=C2)Cl)Cl)NC(=O)C3=CC4=CC=CC=C4S3

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