GSK256073 is a potent and selective agonist of the GPR109A receptor, also known as hydroxy-carboxylic acid receptor 2 (HCA2). With a pEC50 of 7.5 in human HCA2, this orally active compound acts as a full agonist without causing flushing. GSK256073 has demonstrated the ability to acutely enhance glucose homeostasis by inhibiting lipolysis, making it a valuable tool for research into type 2 diabetes mellitus (T2DM) and dyslipidemia.
GSK256073 is a potent and selective agonist of the GPR109A receptor, also known as hydroxy-carboxylic acid receptor 2 (HCA2). With a pEC50 of 7.5 in human HCA2, this orally active compound acts as a full agonist without causing flushing. GSK256073 has demonstrated the ability to acutely enhance glucose homeostasis by inhibiting lipolysis, making it a valuable tool for research into type 2 diabetes mellitus (T2DM) and dyslipidemia.
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