GSK3368715

Catalog No.: A19136

PRMT inhibitor

GSK3368715

GSK3368715 Chemical Structure

CAS NO. 1629013-22-4

GSK3368715 (EPZ019997) is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)).

Availability: In stock

Package Price Qty
1 mg

Regular Price: $500.00

Special Price $400.00

5 mg

Regular Price: $920.00

Special Price $736.00

10 mg

Regular Price: $1,400.00

Special Price $1,120.00

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Biological Activity

GSK3368715 (EPZ019997) is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.28 mL 136.41 mL 272.82 mL
0.5 mM 5.46 mL 27.28 mL 54.56 mL
1 mM 2.73 mL 13.64 mL 27.28 mL
5 mM 0.55 mL 2.73 mL 5.46 mL

*The above data is based on the productmolecular weight 366.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A19136
Actions Inhibitor
CAS No. 1629013-22-4
Formula C20H38N4O2
M. Wt 366.54
Purity >98%
Synonyms GSK 3368715, GSK-3368715
SMILES CNCCN(CC1=CNN=C1C2CCC(COCC)(COCC)CC2)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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