GSK3368715 dihydrochloride

Catalog No.: A21733

PRMT inhibitor

GSK3368715 dihydrochloride

GSK3368715 dihydrochloride Chemical Structure

CAS NO. 1628925-77-8

GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)).

Availability: In stock

Package Price Qty
1 mg
$180.00
5 mg
$540.00
10 mg
$920.00
50 mg
$2,760.00
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Biological Activity

GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50=3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.76 mL 113.78 mL 227.55 mL
0.5 mM 4.55 mL 22.76 mL 45.51 mL
1 mM 2.28 mL 11.38 mL 22.76 mL
5 mM 0.46 mL 2.28 mL 4.55 mL

*The above data is based on the productmolecular weight 439.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21733
Actions Inhibitor
M. Wt 439.46
Formula C20H40Cl2N4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1628925-77-8
Synonyms EPZ019997 dihydrochloride, EPZ-019997, EPZ 019997; GSK-3368715, GSK 3368715
SMILES CNCCN(CC1=CNN=C1C2CCC(COCC)(COCC)CC2)C.Cl.Cl

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