GSK5182
Important Notice: For research use only. We do not sell to patients.
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Important Notice: For research use only. We do not sell to patients.
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Discription | GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα. | ||
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Targets |
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Catalog Num | A19383 |
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Formula | C27H31NO3 |
Molecular Weight | 417.54 |
CAS Number | 877387-37-6 |
SMILES | OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(OCCN(C)C)C=C3 |
Synonyms | GSK 5182, GSK-5182 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 78 mg/mL | |
Water | Insoluble | ||
Ethanol | 78 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 23.95 mL | 119.75 mL | 239.5 mL |
0.5 mM | 4.79 mL | 23.95 mL | 47.9 mL |
1 mM | 2.39 mL | 11.97 mL | 23.95 mL |
5 mM | 0.48 mL | 2.39 mL | 4.79 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2