Biological Activity
GSK5182 is a highly selective inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM and does not interact with other nuclear receptors, including ERRα or ERα.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 23.95 mL | 119.75 mL | 239.5 mL |
0.5 mM | 4.79 mL | 23.95 mL | 47.9 mL |
1 mM | 2.39 mL | 11.97 mL | 23.95 mL |
5 mM | 0.48 mL | 2.39 mL | 4.79 mL |
*The above data is based on the productmolecular weight 417.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A19383 |
---|---|
Actions | Agonist |
M. Wt | 417.54 |
Formula | C27H31NO3 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 877387-37-6 |
Synonyms | GSK 5182, GSK-5182 |
SMILES | OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(OCCN(C)C)C=C3 |
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