GSK8612

Catalog No.: A19438

TBK1 inhibitor

GSK8612

GSK8612 Chemical Structure

CAS NO. 2361659-62-1

GSK8612 is a highly selective and potent Tank-binding Kinase-1 (TBK1) inhibitor, with a pIC50 of 6.8 for recombinant TBK1.

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$140.00
50 mg
$420.00
100 mg
$720.00
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Biological Activity

GSK8612 is a highly selective and potent Tank-binding Kinase-1 (TBK1) inhibitor, with a pIC50 of 6.8 for recombinant TBK1.
In vitro DMSO 92 mg/mL (176.81 mM)
Water Insoluble
Ethanol 6 mg/mL (11.53 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.22 mL 96.09 mL 192.19 mL
0.5 mM 3.84 mL 19.22 mL 38.44 mL
1 mM 1.92 mL 9.61 mL 19.22 mL
5 mM 0.38 mL 1.92 mL 3.84 mL

*The above data is based on the productmolecular weight 520.33. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A19438
Actions Inhibitor
CAS No. 2361659-62-1
Formula C17H17BrF3N7O2S
M. Wt 520.33
Purity >98%
Synonyms GSK-8612; GSK 8612
SMILES NS(C1=CC=C(CNC2=C(Br)C=NC(NC3=CN(CC(F)(F)F)N=C3C)=N2)C=C1)(=O)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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